SCHEMBL6609671

SCHEMBL6609671

Cc1cc(C)nc(Nc2ccc(NC(=O)OC3CC(=O)N(C4Cc5ccccc5C4)C3)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.47
ACHE P22303 4/20 0.46
ALDH1A1 P00352 1/20 0.42
SLC2A1 P11166 4/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
THRB P10828 1/20 0.39
OGG1 O15527 1/20 0.37
TGM2 P21980 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611423 0.87 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL6613611 0.86 ACHE (0.42) BCHEACHEALDH1A1KDM4EHPGD
SCHEMBL6611305 0.86 BCHE (0.59) BCHEACHEALDH1A1RAB9ANPC1
SCHEMBL5843125 0.83 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2
SCHEMBL6611378 0.82 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL6609227 0.81 BCHE (0.55) BCHEACHEALDH1A1RAB9ANPC1
SCHEMBL6611945 0.81 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL6610605 0.81 ACHE (0.49) BCHEACHEALDH1A1MEN1KMT2A
SCHEMBL6610853 0.81 ALOX15 (0.45) BCHEACHEALDH1A1SLC2A1MEN1
SCHEMBL6611127 0.80 NPSR1 (0.49) ALDH1A1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463724-A1 PYRROLIDONE CARBOXAMIDES Actelion Pharmaceuticals Ltd. (CH) 2004-10-06 EP disclosed
WO-2003059905-A1 PYRROLIDONE CARBOXAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2003-07-24 WO disclosed