SCHEMBL6612974

SCHEMBL6612974

O=C1CNC(=O)C2(CCN(c3ccccc3)CC2)N1CCc1c[nH]c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.55
HTR2A P28223 5/20 0.55
HTR1A P08908 5/20 0.55
DRD4 P21917 2/20 0.55
DRD3 P35462 2/20 0.55
SLC6A4 P31645 2/20 0.55
HRH1 P35367 1/20 0.55
HTR2B P41595 1/20 0.55
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTR7 P34969 4/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HTR6 P50406 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6614882 0.89 HTR2A (0.51) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6612040 0.86 DRD3 (0.56) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6610961 0.85 HTR1A (0.59) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6617707 0.84 HTR1A (0.63) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6612983 0.83 HTR1A (0.62) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6611417 0.83 HTR1A (0.62) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6612492 0.82 HTR1A (0.46) DRD2HTR1AKMT2AMAPTLMNA
SCHEMBL6617457 0.81 DRD2 (0.50) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6609843 0.79 CXCR3 (0.49) DRD2HTR2AHTR1ADRD4DRD3
SCHEMBL6012396 0.78 DRD2 (0.44) DRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed