SCHEMBL6613124

SCHEMBL6613124

O=C(NCc1cccs1)c1cc2c(NCc3cnc[nH]3)cccc2s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.48
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 7/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TSHR P16473 3/20 0.42
POLB P06746 2/20 0.42
HTT P42858 2/20 0.42
NPC1 O15118 2/20 0.42
TP53 P04637 1/20 0.42
ADRA1D P25100 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADRA2C P18825 1/20 0.39
MAOB P27338 1/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6757258 0.94 ADRA1A (0.43) ADRA1AALDH1A1KDM4EHSD17B10HPGD
Trifluoroacetic Acid SCHEMBL6760834 0.71 FNTA (0.53)
SCHEMBL17009252 0.64 RAB9A (0.71) ALDH1A1KDM4EHSD17B10HPGDRAB9A
SCHEMBL10837292 0.62 HPGD (0.59) KDM4EHSD17B10HPGDPOLBHTT
SCHEMBL27551588 0.62 ADRA1D (1.00) SMN1; SMN2ADRA1DMAPT
SCHEMBL12265889 0.60 HPGD (0.67) ALDH1A1KDM4EHSD17B10HPGDRAB9A
SCHEMBL31188605 0.60 TAAR1 (0.55) ALDH1A1KDM4ERAB9ASMN1; SMN2TSHR
SCHEMBL4173674 0.60 HPGD (0.68) ALDH1A1KDM4EHPGDRAB9ASMN1; SMN2
SCHEMBL29818326 0.60 HPGD (0.68) ALDH1A1HPGDRAB9ASMN1; SMN2POLB
SCHEMBL28820363 0.60 ALDH1A1 (0.60) ALDH1A1HPGDRAB9ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395581-A2 NOVEL BENZOTHIENYL OR INDOLE DERIVATIVES, PREPARATION AND USE THEREOF AS INHIBITORS OF PRENYL TRANSFERASE PROTEINS PIERRE FABRE MEDICAMENT (FR) 2004-03-10 EP disclosed
WO-2002098852-A2 NOVEL BENZOTHIENYL OR INDOLE DERIVATIVES, AND USE THEREOF AS INHIBITORS OF PRENYL TRANSFERASE PROTEINS PIERRE FABRE MEDICAMENT (FR) 2002-12-12 WO disclosed