SCHEMBL6617416

SCHEMBL6617416

COC(=O)c1cc2cc(NC(=O)OC(C)(C)C)ccc2[nH]1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LEF1 Q9UJU2 1/20 0.74
MMP13 P45452 2/20 0.54
XDH P47989 2/20 0.50
MMP2 P08253 1/20 0.46
TP53 P04637 1/20 0.44
KDM4E B2RXH2 5/20 0.44
RAB9A P51151 6/20 0.43
NPC1 O15118 5/20 0.43
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
PRNP P04156 1/20 0.43
GAA P10253 1/20 0.43
KCNQ2 O43526 1/20 0.43
HPGD P15428 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6619949 0.95 LEF1 (0.81) LEF1MMP13XDHTP53KDM4E
SCHEMBL3031344 0.90 LEF1 (0.61) LEF1MMP13XDHRAB9ANPC1
SCHEMBL3030225 0.88 LEF1 (0.60) LEF1MMP13MMP2TP53KDM4E
SCHEMBL3027522 0.88 MMP13 (0.72) LEF1MMP13MMP2KDM4ERAB9A
SCHEMBL13311254 0.87 LEF1 (0.59) LEF1MMP13MMP2TP53KDM4E
SCHEMBL29830077 0.84 LEF1 (0.67) LEF1MMP13TP53KDM4ERAB9A
SCHEMBL29783677 0.84 FLT3 (0.59) LEF1PDGFRBPDGFRAFLT3
SCHEMBL20742974 0.84 FLT3 (0.59) LEF1PDGFRBPDGFRAFLT3
SCHEMBL7833243 0.83 LEF1 (0.55) LEF1MMP13XDHMMP2TP53
SCHEMBL14138263 0.83 LEF1 (0.55) LEF1MMP13MMP2TP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983248-B1 ANALOGS OF DUOCARMYCIN AND CC-1065 SCRIPPS RESEARCH INST (US) 2004-07-14 EP disclosed
US-6281354-B1 ANTIBIOTICS; ANTITUMOR AGENTS THE SCRIPPS RESEARCH INSTITUTE 2001-08-28 US disclosed
EP-0983248-A4 ANALOGS OF DUOCARMYCIN AND CC-1065 SCRIPPS RESEARCH INST (US) 2000-09-13 EP disclosed
EP-0983248-A1 ANALOGS OF DUOCARMYCIN AND CC-1065 The Scripps Research Institute (US) 2000-03-08 EP disclosed
WO-1998052925-A1 ANALOGS OF DUOCARMYCIN AND CC-1065 THE SCRIPPS RESEARCH INSTITUTE (US) 1998-11-26 WO disclosed