SCHEMBL6621807

SCHEMBL6621807

CC(C)CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)C1CCC(=O)C1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.39
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
CETP P11597 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6620267 0.94 UBE2M (0.36) TACR1SLC6A2SLC6A4CETP
SCHEMBL5215277 0.84 TACR1 (0.40) TACR1
SCHEMBL6621794 0.82 TACR1 (0.49) TACR1
SCHEMBL5212179 0.72 TACR1 (0.37) TACR1
SCHEMBL5729938 0.70 CCR2 (0.49) TACR1
SCHEMBL6957247 0.68 HTT (0.47) TACR1
SCHEMBL3287967 0.67 ALDH1A1 (0.44)
SCHEMBL14169881 0.66 CCR2 (0.40) TACR1CETP
SCHEMBL6056589 0.66 PTGDR2 (0.44)
SCHEMBL6965223 0.62 HTT (0.51) TACR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318811-A4 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2004-07-14 EP disclosed
EP-1318811-A1 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2003-06-18 EP disclosed
WO-2002013824-A1 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2002-02-21 WO disclosed