SCHEMBL6630002

SCHEMBL6630002

CC(C)(C)NS(=O)(=O)c1ccccc1-c1ccc(CN)cc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 18/20 0.57
FEN1 P39748 18/20 0.57
OPRM1 P35372 1/20 0.49
OPRK1 P41145 1/20 0.49
NSD2 O96028 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266847 0.89 ALOX5AP (0.55) ALOX5APFEN1OPRM1OPRK1
SCHEMBL7190899 0.87 ALOX5AP (0.55) ALOX5APFEN1OPRM1OPRK1
SCHEMBL2280981 0.85 ALOX5AP (0.54) ALOX5APFEN1OPRM1OPRK1
SCHEMBL7266374 0.84 OPRM1 (0.54) ALOX5APFEN1OPRM1OPRK1
SCHEMBL6974699 0.83 ALOX5AP (0.53) ALOX5APFEN1OPRM1OPRK1
SCHEMBL890585 0.83 ALOX5AP (0.65) ALOX5APFEN1
SCHEMBL6771873 0.83 EDNRA (0.58) ALOX5APFEN1OPRM1OPRK1
SCHEMBL1968159 0.82 ALOX5AP (0.59) ALOX5APFEN1NSD2
Hydrochloric Acid SCHEMBL6175800 0.82 ALOX5AP (0.64) ALOX5APFEN1NSD2
SCHEMBL6628076 0.81 ALOX5AP (0.59) ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874629-B1 ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2004-05-19 EP disclosed
WO-2003101381-A2 1,2 DIAMIDO CYCLOALKYL SODIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2003-12-11 WO disclosed
US-5939418-A ANTICOAGULANT THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1999-08-17 US disclosed
US-5411980-A Substituted triazolinones, triazolinethiones, and triazolinimines as angiotensin II antagonists MERCK & CO., INC. (US) 1995-05-02 US disclosed