SCHEMBL6630880

SCHEMBL6630880

NC(=O)c1cc(Oc2ccccc2)ccc1N1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.54
HTR1A P08908 3/20 0.51
SLC6A2 P23975 3/20 0.51
SLC6A4 P31645 3/20 0.51
SLC6A3 Q01959 2/20 0.51
MAPK8 P45983 1/20 0.51
MAPK10 P53779 1/20 0.51
SCN9A Q15858 2/20 0.46
SCN4A P35499 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
ALOX15 P16050 1/20 0.45
GFER P55789 1/20 0.45
YWHAG P61981 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6629017 0.89 HTR3A (0.46) LTA4HHTR1AMAPK8MAPK10SCN9A
SCHEMBL6630884 0.80 LTA4H (0.60) LTA4HHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL11908418 0.78 ALDH1A1 (0.59) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL1450313 0.77 NPC1 (0.70) HTR1AKDM4EMAPTHSD17B10NPC1
SCHEMBL16613220 0.77 LTA4H (0.58) LTA4HHTR1AMAPK8MAPK10SCN9A
SCHEMBL11217216 0.76 HSD17B10 (0.53) KDM4EMEN1MAPTTHRBALOX15
Hydrochloric Acid SCHEMBL16597755 0.76 LTA4H (0.56) LTA4HHTR1AMAPK8MAPK10SCN9A
Hydrochloric Acid SCHEMBL27658727 0.76 NPC1 (0.68) HTR1AKDM4EMAPTHSD17B10NPC1
SCHEMBL28881569 0.76 BTK (0.70) LTA4HHTR1ASLC6A4MAPK8MAPK10
SCHEMBL29987229 0.76 BTK (0.70) LTA4HHTR1ASLC6A4MAPK8MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389194-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-02-18 EP disclosed
WO-2002088101-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-07 WO disclosed