SCHEMBL6632646

SCHEMBL6632646

CC(=O)N1CCC[C@H]1C(=O)NC(C(=O)O)C(C)NC(=O)N1CCC2(CC1)C(=O)NCN2c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PLD2 O14939 2/20 0.46
PLD1 Q13393 2/20 0.46
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
SLC18A3 Q16572 1/20 0.45
CALCRL Q16602 1/20 0.45
OPRK1 P41145 4/20 0.44
OPRM1 P35372 3/20 0.44
OPRD1 P41143 2/20 0.44
OPRL1 P41146 2/20 0.44
SLC6A9 P48067 1/20 0.44
HTR2C P28335 1/20 0.44
DRD3 P35462 1/20 0.44
AVPR1A P37288 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5799198 0.86 OPRK1 (0.55) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5950640 0.85 OPRK1 (0.47) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5950573 0.83 OPRK1 (0.47) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5950194 0.82 OPRK1 (0.46) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5950642 0.80 OPRK1 (0.46) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5800244 0.79 CCR5 (0.52) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5802779 0.78 OPRK1 (0.54) PLD2PLD1CTSBCTSSCTSK
SCHEMBL5800621 0.77 CTSB (0.50) PLD2PLD1CTSBCTSSCTSK
SCHEMBL21634299 0.73 HSD17B10 (0.62) SLC18A3OPRK1OPRM1OPRD1OPRL1
SCHEMBL13853705 0.72 OPRK1 (0.58) SLC18A3OPRK1OPRM1OPRD1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1489081-A1 SPIRO DERIVATIVES AND ADHESION MOLECULE INHIBITORS COMPRISING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2004-12-22 EP disclosed