SCHEMBL5800244

SCHEMBL5800244

CC(NC(=O)N1CCC2(CC1)C(=O)NCN2c1ccccc1)C(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.52
CTSB P07858 1/20 0.52
CTSS P25774 1/20 0.52
CTSK P43235 1/20 0.52
OPRK1 P41145 6/20 0.48
OPRM1 P35372 4/20 0.48
OPRD1 P41143 3/20 0.48
OPRL1 P41146 3/20 0.48
SLC6A9 P48067 2/20 0.46
PLD1 Q13393 6/20 0.45
PLD2 O14939 4/20 0.45
HTR2C P28335 1/20 0.45
DRD3 P35462 1/20 0.45
AVPR1A P37288 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5799198 0.90 OPRK1 (0.55) CTSBCTSSCTSKOPRK1OPRM1
SCHEMBL5950765 0.84 ENPP2 (0.50) OPRK1OPRM1OPRD1OPRL1DRD3
SCHEMBL5802422 0.81 NPC1L1 (0.49)
SCHEMBL5802779 0.81 OPRK1 (0.54) CTSBCTSSCTSKOPRK1OPRM1
SCHEMBL5950420 0.81 CCR5 (0.53) CCR5CTSBCTSSCTSKOPRK1
SCHEMBL5800911 0.81 NPC1L1 (0.49) OPRK1OPRM1OPRD1OPRL1
SCHEMBL5800621 0.80 CTSB (0.50) CCR5CTSBCTSSCTSKOPRK1
SCHEMBL6632646 0.79 PLD2 (0.46) CTSBCTSSCTSKOPRK1OPRM1
SCHEMBL318858 0.79 CCR5 (0.75) CCR5OPRK1OPRM1OPRD1OPRL1
SCHEMBL4981531 0.77 SLC6A9 (0.57) CCR5CTSBCTSSCTSKOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329451-B1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES (JP) 2006-08-23 EP disclosed
EP-1489081-A1 SPIRO DERIVATIVES AND ADHESION MOLECULE INHIBITORS COMPRISING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2004-12-22 EP disclosed
EP-1329451-A1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-23 EP disclosed