SCHEMBL6633399

SCHEMBL6633399

CN(C)C(=O)Oc1ccc(N([C@@](C)(C(=O)O)C(=O)[C@H]2NC(C)(C)CS2)S(=O)(=O)c2cccnc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.36
NFE2L2 Q16236 2/20 0.36
ALDH1A1 P00352 4/20 0.34
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 1/20 0.33
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
PTGER2 P43116 2/20 0.30
TSHR P16473 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633018 0.90 KEAP1 (0.34) KEAP1NFE2L2ALDH1A1MAPTKMT2A
SCHEMBL6632994 0.86 HTR1A (0.31)
SCHEMBL6636006 0.85 OXTR (0.32) ALDH1A1KMT2A
SCHEMBL6633881 0.84 ALDH1A1 (0.42) ALDH1A1MAPTGAATSHR
SCHEMBL6633485 0.81
SCHEMBL6634428 0.78 ALDH1A1 (0.33) ALDH1A1MAPTKMT2AGAA
SCHEMBL6632840 0.78 TDP1 (0.32) ALDH1A1MAPTGAA
SCHEMBL6632832 0.78 NCEH1 (0.31)
SCHEMBL6633373 0.77 HSD11B1 (0.33)
SCHEMBL6633653 0.77 HTR1A (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000051-B1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2004-05-19 EP claimed