SCHEMBL6633664

SCHEMBL6633664

COc1ccc2ccc(OC)c(C=CCC(=O)O)c2c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.62
MTNR1B P49286 5/20 0.62
CYP1A2 P05177 3/20 0.48
CYP2C19 P33261 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
HSD17B10 Q99714 2/20 0.47
PTGS1 P23219 1/20 0.47
AKR1C3 P42330 1/20 0.47
AKR1C2 P52895 1/20 0.47
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
CYP2D6 P10635 1/20 0.43
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7741225 0.85 MTNR1A (0.57) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL7741232 0.78 MTNR1A (0.57) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL7741222 0.78 MTNR1A (0.57) MTNR1AMTNR1BCYP1A2CYP2C19CYP3A4
SCHEMBL5227187 0.75 MTNR1A (0.59) MTNR1AMTNR1BCYP1A2CYP2C19CYP2C9
SCHEMBL7741227 0.73 MTNR1A (0.47) MTNR1AMTNR1BHSD17B10PTGS1AKR1C3
SCHEMBL11718070 0.71 KDM4E (0.53) MTNR1AMTNR1BHSD17B10ALDH1A1HPGD
SCHEMBL3914252 0.71 MTNR1A (0.64) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL30692247 0.71 MTNR1A (0.64) MTNR1AMTNR1BHTR2CHTR2B
SCHEMBL2998855 0.70 PAM (0.61) CYP3A4ALDH1A1KDM4E
SCHEMBL2998851 0.70 PAM (0.61) CYP3A4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047664-B1 NOVEL TRICYCLIC COMPOUNDS, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-05-19 EP disclosed