SCHEMBL6645913

SCHEMBL6645913

Cc1ccc(NCCNc2ccc(C)cn2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.53
RAB9A P51151 2/20 0.53
KDM4E B2RXH2 5/20 0.49
CCR1 P32246 1/20 0.46
CCR5 P51681 1/20 0.46
CCR8 P51685 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
ALDH1A1 P00352 5/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
ACKR3 P25106 2/20 0.46
HCAR3 P49019 3/20 0.44
LMNA P02545 1/20 0.44
PKM P14618 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADRA2A P08913 3/20 0.44
ADRA2B P18089 3/20 0.44
ADRA2C P18825 3/20 0.44
NOS3 P29474 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12830407 0.92 MAPT (0.47) MAPTRAB9AKDM4ECCR1CCR5
SCHEMBL10293613 0.90 HCAR3 (0.57) MAPTRAB9AKDM4ECCR1CCR5
SCHEMBL10737266 0.89 HRH3 (0.47) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL12832042 0.88 RAB9A (0.52) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL13103613 0.88 RAB9A (0.47) MAPTRAB9AKDM4ECCR1CCR5
SCHEMBL12832443 0.87 CYP2C19 (0.56) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL10604098 0.86 HCAR3 (0.59) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL22197869 0.86 CASP2 (0.43) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL12060 0.85 CYP2C19 (0.57) MAPTRAB9AKDM4EALDH1A1GAA
SCHEMBL11563180 0.85 ALDH1A1 (0.51) MAPTRAB9AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087963-B1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORP (US) 2004-08-25 EP disclosed