SCHEMBL6651356

SCHEMBL6651356

CN(C)CCOc1cccc(Cc2ccnn2C)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
DRD5 P21918 1/20 0.44
HTR7 P34969 3/20 0.40
HTR1B P28222 1/20 0.40
HRH1 P35367 2/20 0.38
P2RX7 Q99572 1/20 0.38
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
UTS2R Q9UKP6 2/20 0.35
KAT2B Q92831 1/20 0.35
NR4A2 P43354 1/20 0.35
LMNA P02545 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6892797 0.88 DRD2 (0.58) DRD2DRD1DRD4DRD5HTR7
SCHEMBL6651166 0.83 KDM4E (0.38) DRD2DRD1DRD4DRD5HTR7
SCHEMBL6650105 0.81 NR4A2 (0.42) DRD2DRD1DRD4DRD5P2RX7
Citric Acid SCHEMBL8657218 0.75 KDM4E (0.70) DRD2DRD1DRD4DRD5HRH1
SCHEMBL4303080 0.73 HTR7 (0.36) DRD2DRD1DRD4DRD5HTR7
SCHEMBL4909282 0.73 KAT2B (0.34) DRD2DRD1DRD4DRD5HTR7
SCHEMBL6650106 0.72 P2RX7 (0.46) DRD4P2RX7KDM4EALDH1A1LMNA
SCHEMBL19471246 0.72 P2RX7 (0.38) P2RX7KDM4EALDH1A1LMNA
SCHEMBL7755878 0.72 LTA4H (0.56) CHRNB2CHRNA4
SCHEMBL5599334 0.70 ADRB2 (0.35) DRD2DRD1DRD4DRD5HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed