SCHEMBL6653211

SCHEMBL6653211

O=c1oc(Cl)ccc1Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTRC Q99895 6/20 1.00
GPR55 Q9Y2T6 7/20 0.48
CNR2 P34972 3/20 0.48
CEL P19835 4/20 0.46
NR1H2 P55055 1/20 0.41
MEN1 O00255 1/20 0.40
ELANE P08246 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27429798 0.69 CTRC (0.53) CTRCGPR55CNR2NR1H2
SCHEMBL29709847 0.68 GPR55 (0.68) CTRCGPR55
SCHEMBL19331106 0.68 GPR55 (0.68) CTRCGPR55
SCHEMBL28412953 0.67 ELANE (0.53) CTRCNR1H2ELANE
SCHEMBL8098213 0.66 CALM1 (0.55) CTRCGPR55CNR2
SCHEMBL972711 0.65 CALM1 (0.69) MEN1KMT2A
SCHEMBL11403614 0.65 CALM1 (0.52) CTRCNR1H2MEN1KMT2A
SCHEMBL4423210 0.65 SIGMAR1 (0.53) CTRCMEN1KMT2A
SCHEMBL2861971 0.64 CTRC (0.47) CTRCNR1H2MEN1KMT2A
SCHEMBL160386 0.64 BCL2 (0.48) CTRCGPR55CNR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1323715-B1 Inhibitors of cholesterol esterase UNIV NEW MEXICO (US) 2004-06-30 EP disclosed
EP-0975617-B1 INHIBITORS OF CHOLESTEROL ESTERASE UNIV NEW MEXICO (US) 2003-11-05 EP disclosed
EP-1323715-A1 Inhibitors of cholesterol esterase The University of New Mexico (US) 2003-07-02 EP disclosed
EP-0975617-A4 INHIBITORS OF CHOLESTEROL ESTERASE UNIV NEW MEXICO (US) 2000-09-13 EP disclosed
US-6114545-A Inhibitors of cholesterol esterase UNIVERSITY OF NEW MEXICO (US) 2000-09-05 US disclosed
US-6034255-A Inhibitors of cholesterol esterase UNIVERSITY OF NEW MEXICO (US) 2000-03-07 US disclosed
EP-0975617-A1 INHIBITORS OF CHOLESTEROL ESTERASE The University of New Mexico (US) 2000-02-02 EP disclosed
US-5942631-A Inhibitors of cholesterol esterase UNIVERSITY OF NEW MEXICO (US) 1999-08-24 US disclosed
WO-1998046585-A1 INHIBITORS OF CHOLESTEROL ESTERASE THE UNIVERSITY OF NEW MEXICO (US) 1998-10-22 WO disclosed