SCHEMBL6653306

SCHEMBL6653306

CC(C)=CCOc1ccc(C(=O)O)c(OCC=C(C)C)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.60
HPGD P15428 2/20 0.60
MEN1 O00255 1/20 0.60
NR1I2 O75469 1/20 0.60
LMNA P02545 1/20 0.60
PGR P06401 1/20 0.60
ADRB2 P07550 1/20 0.60
ADRB1 P08588 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
CNR1 P21554 1/20 0.60
TBXA2R P21731 1/20 0.60
SLC6A2 P23975 1/20 0.60
AGTR1 P30556 1/20 0.60
ADRA1A P35348 1/20 0.60
OPRD1 P41143 1/20 0.60
OPRK1 P41145 1/20 0.60
BLM P54132 1/20 0.60
SLC6A3 Q01959 1/20 0.60
KMT2A Q03164 1/20 0.60
ALOX5 P09917 4/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28964412 0.91 ALOX5 (0.55) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL6652397 0.89 ALOX5 (0.53) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL5384385 0.89 MAOB (0.55) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL3901893 0.89 ALOX5 (0.58) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL6652010 0.88 ALOX15 (0.56) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL6652005 0.88 ALOX15 (0.56) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL28948144 0.86 MAOB (0.49) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL28948158 0.85 HPGD (0.45) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL28948098 0.85 TSHR (0.54) MAPTHPGDMEN1NR1I2LMNA
SCHEMBL9364600 0.84 MEN1 (0.70) MAPTHPGDMEN1NR1I2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0875501-B1 Alkylenediamine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO CO LTD (JP) 2004-06-16 EP disclosed
EP-0802196-B1 Alkylenediamine derivatives as drugs for the treatment of ulcers and the inhibition of Helicobacter pylori SHISEIDO CO LTD (JP) 2001-08-29 EP disclosed
US-6043243-A Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO CO., LTD. (JP) 2000-03-28 US disclosed
US-6001880-A DISUBSTITUTED N-(2-DIALKYLAMINOETHYL)BENZAMIDE DERIVATIVES OF GIVEN FORMULA; ANTIBACTERIAL ACTIVITY AGAINST HELICOBACTER PYROLI, ADMINISTERING FOR THE PREVENTION OR CURE OF PEPTIC ULCERS SHISEIDO CO., LTD. (JP) 1999-12-14 US disclosed
US-5925667-A INHIBITS GROWTH OF HELICOBACTER PYLORI SHISEIDO CO., LTD. (JP) 1999-07-20 US disclosed
EP-0875501-A2 Alkylenediamine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1998-11-04 EP disclosed
EP-0869118-A1 Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1998-10-07 EP disclosed
US-5814634-A PEPTIC ULCERS, GASTRIC ULCERS SHISEIDO CO. LTD. (JP) 1998-09-29 US disclosed
EP-0802196-A1 Alkylenediamine derivative, antiulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1997-10-22 EP disclosed