SCHEMBL6660147

SCHEMBL6660147

CC(C)(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N(C#N)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSS P25774 14/20 0.47
CTSK P43235 12/20 0.47
CTSL P07711 3/20 0.41
CTSB P07858 2/20 0.41
PTPN1 P18031 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6657069 0.95 CTSS (0.48) CTSSCTSKCTSLCTSB
SCHEMBL6048161 0.85 CTSS (0.46) CTSSCTSKCTSLCTSB
SCHEMBL5696941 0.74 PPARG (0.43) CTSSCTSKCTSLCTSB
SCHEMBL6048166 0.73 CTSK (0.38) CTSSCTSKCTSLCTSBKMT2A
SCHEMBL24856016 0.72 JAK3 (0.51) CTSSCTSKCTSLCTSB
SCHEMBL20027759 0.72 JAK3 (0.51) CTSSCTSKCTSLCTSB
SCHEMBL24325842 0.72 JAK3 (0.51) CTSSCTSKCTSLCTSB
SCHEMBL2713175 0.71 CTSK (0.37) CTSSCTSKCTSLCTSBKMT2A
SCHEMBL1360500 0.70 CTSK (0.51) CTSSCTSKCTSLCTSBKMT2A
SCHEMBL66303 0.70 CTSK (0.51) CTSSCTSKCTSLCTSBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1434769-A2 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-07-07 EP disclosed
WO-2003029200-A2 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2003-04-10 WO disclosed