SCHEMBL6661408

SCHEMBL6661408

COC1=C(OC)C(=O)C(c2ccc(C(=O)Nc3ccc(C(F)(F)F)cc3)c(-c3ccccc3)c2C)=C(C)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR27 Q9NS67 3/20 0.44
AVPR2 P30518 2/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
PTGS1 P23219 1/20 0.42
MAOB P27338 1/20 0.41
SMO Q99835 4/20 0.40
GAA P10253 2/20 0.40
POLB P06746 1/20 0.40
MTTP P55157 4/20 0.40
APOB P04114 3/20 0.40
CISD2 Q8N5K1 1/20 0.40
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
HTR1A P08908 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859183 0.89 MAPT (0.49) NPC1RAB9ASMN1; SMN2GMNNLMNA
SCHEMBL5860306 0.80 SMO (0.44) NPC1RAB9ASMN1; SMN2PTGS1SMO
SCHEMBL5860276 0.79 PDE4B (0.43) RAB9ASMN1; SMN2POLBGMNNLMNA
SCHEMBL5860337 0.78 APOB (0.44) SMOMTTPAPOB
SCHEMBL5859192 0.78 PSMD14 (0.51) RAB9AGAAPOLBLMNA
SCHEMBL5862249 0.75 MTTP (0.45) GPR27AVPR2SMN1; SMN2GAAPOLB
SCHEMBL5860012 0.75 PPARA (0.46) GPR27AVPR2NPC1RAB9ASMN1; SMN2
SCHEMBL5859923 0.75 MAPT (0.49) SMN1; SMN2LMNANPSR1
SCHEMBL5859855 0.73 NPC1 (0.51) NPC1RAB9AMAOBGAAPOLB
SCHEMBL5860301 0.71 SMO (0.44) SMN1; SMN2SMOMTTPAPOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed