SCHEMBL5860306

SCHEMBL5860306

COC1=C(OC)C(=O)C(c2c(C)ccc(C(=O)Nc3ccc(C(F)(F)F)cc3)c2-c2ccncc2)=C(C)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 5/20 0.44
APOB P04114 6/20 0.43
MTTP P55157 6/20 0.43
TRPV1 Q8NER1 4/20 0.42
BRAF P15056 1/20 0.41
PTGS1 P23219 1/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
KIT P10721 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
NPC1 O15118 1/20 0.41
GMNN O75496 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5860337 0.86 APOB (0.44) SMOAPOBMTTPTRPV1BRAF
SCHEMBL6661408 0.80 GPR27 (0.44) SMOAPOBMTTPPTGS1LMNA
SCHEMBL5859183 0.80 MAPT (0.49) TRPV1LMNAMAPTNPC1GMNN
SCHEMBL5860301 0.79 SMO (0.44) SMOAPOBMTTPMAPTJAK2
SCHEMBL5859923 0.78 MAPT (0.49) TRPV1BRAFLMNAMAPTKIT
SCHEMBL5859049 0.77 ROCK1 (0.47) MAPTMAPK1TP53CYP3A4CYP2C9
SCHEMBL5859281 0.76 CYP3A4 (0.48) BRAFLMNAMAPTJAK2TYK2
SCHEMBL5860289 0.73 PPARA (0.43) APOBMTTPLMNAMAPTMAPK1
SCHEMBL5860280 0.73 CYP46A1 (0.42) LMNACYP2C9HTTSMN1; SMN2NPSR1
SCHEMBL5859178 0.70 MAPT (0.48) TRPV1LMNAMAPTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed