SCHEMBL6663843

SCHEMBL6663843

CC(=O)N1CCc2c1cc(C)c(NC(=O)c1cc(C(F)(F)F)ccc1-c1ccccc1)c2C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 4/20 0.44
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
MTTP P55157 3/20 0.39
KDM4E B2RXH2 1/20 0.38
SLC6A9 P48067 1/20 0.38
NPY5R Q15761 4/20 0.37
APOB P04114 2/20 0.37
TRPV4 Q9HBA0 1/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FABP4 P15090 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6800720 0.91 KDM4E (0.47) NOTUMKMT2AMTTPKDM4EAPOB
SCHEMBL6667054 0.86 SORT1 (0.40)
SCHEMBL6665293 0.81 SORT1 (0.40) MTTPAPOBTRPV4
SCHEMBL6669985 0.80 PARP10 (0.40) MTTPAPOBHCRTR1HCRTR2FABP4
SCHEMBL6667492 0.79 NOTUM (0.60) NOTUMTSHRMTTPAPOBUSP2
SCHEMBL5111860 0.76 MTTP (0.40) TSHRMEN1POLBKMT2AMTTP
SCHEMBL6801395 0.71 SMO (0.47) MTTPKDM4EAPOBLMNAGAA
SCHEMBL14288688 0.70 MTTP (0.52) KMT2AMTTPKDM4EAPOBLMNA
SCHEMBL6809331 0.69 MTTP (0.46) MTTPKDM4EAPOBGAA
SCHEMBL6804769 0.69 MTTP (0.62) NOTUMMTTPKDM4EAPOBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383760-A1 BIARYLCARBOXAMIDE COMPOUNDS AS APOLIPOPROTEIN B INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-28 EP disclosed
WO-2002090347-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-14 WO disclosed