SCHEMBL6671405

SCHEMBL6671405

CN(Cc1ccc(Cl)cc1)C(=O)c1n[nH]c2ccc(C#CCO)cc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
NR1H4 Q96RI1 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
ITK Q08881 2/20 0.34
TTK P33981 1/20 0.34
HAT1 O14929 1/20 0.34
EP300 Q09472 1/20 0.34
MAPK14 Q16539 1/20 0.34
CNR1 P21554 1/20 0.33
PIN1 Q13526 1/20 0.33
GRIN1 Q05586 1/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6672009 0.93 HSP90AA1 (0.39) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL7483549 0.87 HSP90AA1 (0.44) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL7014028 0.85 ALDH1A1 (0.37) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL6672645 0.83 HSP90AA1 (0.42) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL6667497 0.83 HSP90AA1 (0.41) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL7475445 0.82 HSP90AA1 (0.44) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL7843694 0.82 GAA (0.46) ALDH1A1HTTGAA
SCHEMBL6672675 0.79 NR1H4 (0.40) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL6667774 0.77 CHEK1 (0.46) HSP90AA1NR1H4NPC1RAB9AALDH1A1
SCHEMBL7834375 0.76 GABRA1 (0.39) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265873-A2 4-OXO-1,4-DIHYDRO-3-CINNOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-12-18 EP claimed
WO-2001070706-A2 4-OXO-1,4-DIHYDRO-3-CINNOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-09-27 WO claimed
WO-2004019940-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO disclosed