SCHEMBL7014028

SCHEMBL7014028

CN(Cc1ccc(Cl)cc1)C(=O)c1n[nH]c2ncc(C#CCO)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
EGLN1 Q9GZT9 5/20 0.36
HSP90AA1 P07900 1/20 0.36
NR1H4 Q96RI1 1/20 0.35
NPC1 O15118 1/20 0.35
MAP3K20 Q9NYL2 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
MAPK14 Q16539 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6671405 0.85 HSP90AA1 (0.40) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL7014636 0.83 RAB9A (0.38) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL7015761 0.83 ALDH1A1 (0.41) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL6672009 0.78 HSP90AA1 (0.39) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL6672675 0.78 NR1H4 (0.40) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL7007040 0.77 PDE1B (0.45) RAB9ANR1H4NPC1
SCHEMBL7483549 0.76 HSP90AA1 (0.44) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL6672645 0.72 HSP90AA1 (0.42) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL7015592 0.72 HSP90AA1 (0.40) ALDH1A1HTTRAB9AHSP90AA1NR1H4
SCHEMBL6672672 0.72 NR1H4 (0.34) HSP90AA1NR1H4NPC1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1301493-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-04-16 EP claimed
WO-2002004444-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-01-17 WO claimed