SCHEMBL6672415

SCHEMBL6672415

Cc1c(O)ccc(C[C@@H](C(=O)O)N(C)C)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.39
PGR P06401 2/20 0.39
NR3C2 P08235 2/20 0.39
FNTA P49354 3/20 0.35
FNTB P49356 3/20 0.35
HTT P42858 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 2/20 0.33
PPARG P37231 1/20 0.33
TACR1 P25103 1/20 0.33
KDM6B O15054 1/20 0.33
MAPK1 P28482 1/20 0.32
TYR P14679 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
EGFR P00533 1/20 0.32
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673758 0.86 NR3C1 (0.38) NR3C1PGRNR3C2FNTAFNTB
SCHEMBL11593932 0.85 NCEH1 (0.34) HTTMAPTALDH1A1PPARGTACR1
SCHEMBL3450569 0.85 NCEH1 (0.34) HTTMAPTALDH1A1PPARGTACR1
SCHEMBL7941005 0.85 NCEH1 (0.34) HTTMAPTALDH1A1PPARGTACR1
Hydrochloric Acid SCHEMBL11591299 0.84 ALDH1A1 (0.36) HTTMAPTALDH1A1PPARGTACR1
SCHEMBL6671785 0.77 ESR1 (0.40) NR3C1PGRNR3C2HTTMAPT
SCHEMBL5324040 0.77 KDM4E (0.54) FNTAFNTBMAPTALDH1A1KDM4E
SCHEMBL5324035 0.77 KDM4E (0.54) FNTAFNTBMAPTALDH1A1KDM4E
SCHEMBL7277625 0.77 PCNA (0.38) HTTPPARG
SCHEMBL38894 0.76 ESR1 (0.46) NR3C1PGRNR3C2HTTTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004026293-A2 HEMIASTERLIN DERIVATIVES FOR TREATING RESISTANT TUMORS WYETH HOLDINGS CORPORATION (US) 2004-04-01 WO disclosed