SCHEMBL6673752

SCHEMBL6673752

N=C(N)NNCCCC=O

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.36
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6674188 0.87
SCHEMBL261594 0.78
SCHEMBL27780414 0.74 HIF1A (0.39) HIF1ATSHR
Biguanide SCHEMBL28148706 0.73 HIF1A (0.50) HIF1ATSHR
SCHEMBL436282 0.72 ALOX15 (0.47) HIF1ATSHR
Glutaral SCHEMBL28202030 0.71 HIF1A (0.62) HIF1ATSHR
SCHEMBL3166180 0.71
SCHEMBL9539681 0.71 LMNA (0.40) TSHR
SCHEMBL5497459 0.71 MEN1 (0.50) HIF1ATSHR
SCHEMBL7283602 0.71 MEN1 (0.50) HIF1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0627925-B1 TRYPSIN INHIBITORS DENDREON CORP (US) 2004-09-29 EP disclosed
US-5714580-A PROTECTING ALDEHYDE OF AMINOALDEHYDE (I.E. ARGININAL) WITH 4-(DIARYLMETHYL)-SEMICARBAZIDE FOR SUBSEQUENT PEPTIDE ALDEHYDE SYNTHESIS CORVAS INTERNATIONAL, INC. (US) 1998-02-03 US disclosed
EP-0627925-A4 TRYPSIN INHIBITORS. CORVAS INT INC (US) 1997-07-30 EP disclosed
US-5534498-A TREATMENT OF PANCREATITIS CORVAS INTERNATIONAL, INC. (US) 1996-07-09 US disclosed
EP-0627925-A1 TRYPSIN INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1994-12-14 EP disclosed
WO-1993014779-A1 TRYPSIN INHIBITORS CORVAS INTERNATIONAL, INC. (US) 1993-08-05 WO disclosed