SCHEMBL6675758

SCHEMBL6675758

CCOC(=O)OC1Nc2cc(Cl)cc(Cl)c2C2C=CCC12.O=C(O)OC1Nc2cc(Cl)cc(Cl)c2C2C=CCC12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAPDH P04406 3/20 0.56
HSPA1A P0DMV8 2/20 0.56
HSPA8 P11142 2/20 0.56
MEN1 O00255 6/20 0.39
POLB P06746 6/20 0.39
KMT2A Q03164 6/20 0.39
L3MBTL1 Q9Y468 4/20 0.39
PTPN7 P35236 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
NR4A1 P22736 2/20 0.39
BLM P54132 2/20 0.39
PLA2G1B P04054 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MASP2 O00187 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6214303 0.96 GAPDH (0.57) GAPDHHSPA1AHSPA8MEN1POLB
SCHEMBL6214848 0.90 GAPDH (0.68) GAPDHHSPA1AHSPA8MEN1POLB
SCHEMBL6085506 0.79 GAPDH (0.69) GAPDHHSPA1AHSPA8MEN1POLB
SCHEMBL6217839 0.78 CDC25B (0.57) GAPDHHSPA1AHSPA8MEN1POLB
SCHEMBL6211796 0.76 GAPDH (0.35) GAPDHHSPA1AHSPA8
SCHEMBL6087749 0.73 HSPA1A (1.00) GAPDHHSPA1AHSPA8MEN1POLB
SCHEMBL6951562 0.71 CYP2C9 (0.37)
SCHEMBL6217832 0.71 MAPK1 (0.33)
SCHEMBL6214662 0.70 POLB (0.34) MEN1POLBKMT2AL3MBTL1TDP1
SCHEMBL6217040 0.70 CDC25B (0.68) GAPDHHSPA1AHSPA8MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470110-A2 METHOD FOR THE PRODUCTION OF SUBSTITUTED 1,2,3,4-TETRAHYDROQUINOLINE-2-CARBOXYLIC ACIDS Grünenthal GmbH (DE) 2004-10-27 EP disclosed
WO-2003062202-A2 METHOD FOR THE PRODUCTION OF SUBSTITUTED 1,2,3,4-TETRAHYDROISOQUINOLINE-2-CARBOXYLIC ACIDS Grünenthal GmbH (DE) 2003-07-31 WO disclosed