SCHEMBL6676891

SCHEMBL6676891

COc1c(C(C)(C)C)cc(C(C)(C)C)cc1C(C)(C)Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.42
RXRA P19793 2/20 0.40
PPARG P37231 2/20 0.40
RARG P13631 1/20 0.40
PTGS1 P23219 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TNFRSF1A P19438 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
DHFR P00374 1/20 0.36
TP53 P04637 2/20 0.34
LMNA P02545 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2947022 0.91 PTGS2 (0.47) PTGS2RXRAPPARGRARGPTGS1
SCHEMBL6672713 0.83 CA1 (0.55) PTGS2PTGS1ALDH1A1TSHRTDP1
SCHEMBL6673542 0.83 ALDH1A1 (0.45) PTGS2PTGS1ALDH1A1TSHRTDP1
SCHEMBL6673577 0.82 PTGS2 (0.41) PTGS2PTGS1ALDH1A1TSHRTDP1
SCHEMBL3770921 0.82 CA2 (0.42) PTGS2RXRAPPARGRARGPTGS1
SCHEMBL14817161 0.81 RARG (0.40) PTGS2RXRAPPARGRARGPTGS1
SCHEMBL13688744 0.81 ALDH1A1 (0.42) PTGS2RXRAPPARGRARGPTGS1
SCHEMBL10019863 0.79 CYP3A4 (0.42) PTGS2RXRAPPARGRARGALDH1A1
SCHEMBL4297642 0.78 ALOX15 (0.46) PTGS2RXRAPPARGRARGALDH1A1
SCHEMBL12706039 0.78 RARG (0.39) PTGS2RXRAPPARGRARGPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0963990-B1 PROCESS FOR PRODUCING CYCLOPENTADIENYL METAL SALTS AND PROCESS FOR PRODUCING CYCLOPENTADIENE DERIVATIVES BY UTILIZING THE SAME SUMITOMO CHEMICAL CO (JP) 2004-10-06 EP disclosed
US-6197990-B1 REACTING CYCLOPENTADIENE AND METAL HYDRIDE IN PRESENCE OF AMINE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-03-06 US disclosed
EP-0963990-A1 PROCESS FOR PRODUCING CYCLOPENTADIENYL METAL SALTS AND PROCESS FOR PRODUCING CYCLOPENTADIENE DERIVATIVES BY UTILIZING THE SAME SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-12-15 EP disclosed