SCHEMBL6677282

SCHEMBL6677282

CCNC(=NC)Nc1cccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1C

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
BCHE P06276 1/20 0.32
NLRP3 Q96P20 1/20 0.32
BTK Q06187 1/20 0.32
GRM2 Q14416 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
NCOR2 Q9Y618 1/20 0.31
TSHR P16473 1/20 0.31
CACNA1C Q13936 1/20 0.30
SCN5A Q14524 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7242006 0.89 GPR35 (0.38) POLBLMNAHTTALDH1A1GAA
SCHEMBL6676761 0.85 POLB (0.35) POLBLMNAHTTALDH1A1GAA
SCHEMBL7247906 0.81 LMNA (0.34) POLBLMNAHTTALDH1A1GAA
SCHEMBL6677510 0.81 LMNA (0.33) POLBLMNAHTTALDH1A1GAA
SCHEMBL6676767 0.80 CACNA1C (0.43) POLBLMNAHTTALDH1A1NLRP3
SCHEMBL6674712 0.79 ALDH1A1 (0.36) POLBLMNAHTTALDH1A1GAA
SCHEMBL6674967 0.79 GRM2 (0.38) GAAGRM2HDAC3HDAC1HDAC2
SCHEMBL6680745 0.78 GAA (0.33) POLBLMNAHTTALDH1A1GAA
SCHEMBL6677280 0.78 LMNA (0.34) POLBLMNAHTTALDH1A1BCHE
SCHEMBL6676005 0.76 LMNA (0.33) POLBLMNAHTTALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed