SCHEMBL6677458

SCHEMBL6677458

COc1c(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)cccc1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
HTT P42858 1/20 0.41
NR1D1 P20393 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA2 P00918 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
SNCA P37840 1/20 0.38
LMNA P02545 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876745 0.88 ALDH1A1 (0.42) ALDH1A1HTTNR1D1POLBRAB9A
SCHEMBL7872378 0.86 ALDH1A1 (0.41) ALDH1A1HTTNR1D1POLBRAB9A
SCHEMBL6676029 0.85 TDP1 (0.46) ALDH1A1HTTNR1D1NPSR1POLB
SCHEMBL283204 0.84 SMN1; SMN2 (0.42) ALDH1A1HTTNR1D1NPSR1POLB
SCHEMBL6679943 0.84 NR1D1 (0.40) ALDH1A1HTTNR1D1NPSR1RAB9A
SCHEMBL6676172 0.81 KMT2A (0.38) ALDH1A1HTTPOLBSNCALMNA
SCHEMBL6677867 0.79 KDM4E (0.36) ALDH1A1HTTPOLBRAB9ALMNA
SCHEMBL1625905 0.77 BMP1 (0.47) ALDH1A1NR1D1POLBRAB9ATDP1
SCHEMBL1627019 0.77 TSHR (0.44) ALDH1A1NR1D1MAPTTSHR
SCHEMBL5191594 0.76 SNCA (0.49) ALDH1A1NR1D1SNCATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed