SCHEMBL6679083

SCHEMBL6679083

CCN(C(N)=NC(=O)OC(C)(C)C)c1ccc(CNC(=O)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.47
HDAC6 Q9UBN7 5/20 0.47
NR1H2 P55055 1/20 0.46
F2 P00734 2/20 0.44
HDAC3 O15379 6/20 0.44
RAB9A P51151 2/20 0.44
LMNA P02545 1/20 0.44
HDAC2 Q92769 3/20 0.42
EPHX2 P34913 2/20 0.42
NR1H4 Q96RI1 2/20 0.42
NPC1 O15118 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679124 0.89 NR1H4 (0.44) HDAC1HDAC6NR1H2RAB9ALMNA
SCHEMBL6676118 0.78 CA2 (0.47) RAB9ALMNANPC1
SCHEMBL6679078 0.75 NR1H2 (0.50) HDAC1HDAC6NR1H2HDAC3RAB9A
SCHEMBL6685807 0.73 CYP2D6 (0.42)
SCHEMBL6680479 0.73 CYP2C9 (0.39) HDAC1LMNA
SCHEMBL7988109 0.72 GRIN2D (0.49) RAB9ALMNA
SCHEMBL19639298 0.72 NR1H2 (0.49) HDAC1HDAC6NR1H2HDAC3RAB9A
SCHEMBL28966161 0.72 HDAC1 (0.52) HDAC1HDAC6NR1H2HDAC3RAB9A
SCHEMBL6676958 0.71 KDM4E (0.36) HDAC1RAB9ANPC1
SCHEMBL6678219 0.70 SIGMAR1 (0.41) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed