SCHEMBL6681642

SCHEMBL6681642

NS(=O)(=O)c1ccc(-c2ccncc2)c(-c2nccs2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.44
CA2 P00918 5/20 0.41
CA9 Q16790 4/20 0.41
ENPP3 O14638 1/20 0.41
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
IKBKE Q14164 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
CA1 P00915 3/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
CA12 O43570 2/20 0.39
PTGS1 P23219 2/20 0.38
PTGS2 P35354 2/20 0.38
SCN9A Q15858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6623867 0.89 PDPK1 (0.49) LRRK2CA2CA9ENPP3CA1
SCHEMBL27997605 0.89 CA2 (0.43) LRRK2CA2CA9ENPP3CA1
SCHEMBL6624142 0.87 CA2 (0.44) LRRK2CA2CA9ENPP3IKBKB
SCHEMBL20899926 0.83 CA2 (0.45) CA2CA9ENPP3CA1CA12
SCHEMBL20899969 0.78 CA2 (0.51) CA2CA9CA1CA12PTGS2
SCHEMBL6681646 0.76 GABRA1 (0.41) LRRK2CA2CA9ENPP3IKBKB
SCHEMBL31345785 0.75 LOXL2 (0.56) CA2CA9ENPP3CA1CA12
SCHEMBL5693321 0.74 CA2 (0.41) LRRK2CA2CA9ENPP3CA1
SCHEMBL27944286 0.73 CA2 (0.55) CA2CA9ENPP3CA1CA12
Hydrochloric Acid SCHEMBL20899879 0.73 CA2 (0.40) LRRK2CA2CA9ENPP3CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461325-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP disclosed
WO-2003043999-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO disclosed