SCHEMBL6685583

SCHEMBL6685583

Cc1[nH]c2ccc(CCN(C3CCCCC3)S(C)(=O)=O)cc2c1C(=O)OC(C)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MDM2 Q00987 1/20 0.36
HTT P42858 2/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
LMNA P02545 3/20 0.35
SMYD2 Q9NRG4 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPK1 P28482 1/20 0.33
SLC6A3 Q01959 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6316780 0.90 SIGMAR1 (0.41) MEN1KMT2AMAPTALDH1A1MDM2
SCHEMBL6315618 0.83 ALOX5 (0.39) MEN1KMT2AMAPTALDH1A1MDM2
SCHEMBL6692790 0.83 HTT (0.36) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL6321200 0.82 SIGMAR1 (0.44) MAPTALDH1A1MDM2LMNASMN1; SMN2
SCHEMBL6317151 0.80 KMT2A (0.36) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL6316011 0.80 SLC6A3 (0.40) MDM2SLC6A3
SCHEMBL6316297 0.80 MAPK14 (0.40) MEN1KMT2AMAPTALDH1A1MDM2
SCHEMBL6316014 0.80 SIGMAR1 (0.44) LMNASMN1; SMN2SIGMAR1
SCHEMBL6316794 0.79 LMNA (0.39) MEN1KMT2AMAPTALDH1A1MDM2
SCHEMBL6316049 0.79 SIGMAR1 (0.45) LMNASMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377549-A1 FUNCTIONALIZED HETEROCYCLES AS MODULATORS OF CHEMOKINE RECEPTOR FUNCTION AND METHODS OF USE THEREFOR Millennium Pharmaceuticals, Inc. (US) 2004-01-07 EP disclosed
WO-2002072549-A1 FUNCTIONALIZED HETEROCYCLES AS MODULATORS OF CHEMOKINE RECEPTOR FUNCTION AND METHODS OF USE THEREFOR MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-09-19 WO disclosed