SCHEMBL6687083

SCHEMBL6687083

CCCCNC(=O)Nc1cc(C(N)=O)ccc1N1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
CNR1 P21554 2/20 0.53
CNR2 P34972 2/20 0.53
MEN1 O00255 2/20 0.53
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 2/20 0.45
LMNA P02545 3/20 0.44
TP53 P04637 2/20 0.44
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
EPHX2 P34913 1/20 0.42
OPRD1 P41143 3/20 0.42
OPRM1 P35372 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
NPY2R P49146 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968717 1.00 KMT2A (0.53) KMT2ACNR1CNR2MEN1ALDH1A1
SCHEMBL6698122 0.86 KMT2A (0.51) KMT2ACNR1CNR2MEN1ALDH1A1
SCHEMBL29968530 0.86 MAPT (0.58) KMT2AMEN1MAPTLMNATP53
SCHEMBL6687109 0.86 MAPT (0.58) KMT2AMEN1MAPTLMNATP53
SCHEMBL27126152 0.84 KMT2A (0.47) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL29968317 0.84 KMT2A (0.47) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL6695115 0.84 KMT2A (0.47) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL29968131 0.83 MAPT (0.51) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL6686127 0.83 MAPT (0.51) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL6692823 0.82 MAPT (0.47) KMT2AALDH1A1MAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040235855-A1 Phospholipase C inhibitors for use in treating inflammatory disorders JANSSEN PHARMACEUTICA, N.V. (BE) 2004-11-25 US claimed
WO-2004087685-A2 PHOSPHOLIPASE C INHIBITORS FOR USE IN TREATING INFLAMMATORY DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 2004-10-14 WO claimed
US-20250017878-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY CHRONIC AIRWAY THERAPEUTICS LTD (AU) 2025-01-16 US disclosed
CN-117999073-A Use of nadolol to treat chronic obstructive pulmonary disease by blocking the inhibitor protein-2 pathway 慢性呼吸道治疗有限公司 2024-05-07 CN disclosed
EP-4304717-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY Chronic Airway Therapeutics Limited (AU) 2024-01-17 EP disclosed
WO-2004087685-A2 PHOSPHOLIPASE C INHIBITORS FOR USE IN TREATING INFLAMMATORY DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 2004-10-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250017878-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY ARRB1, ADRB2, ADRB1 KMT2A 3828/4885CNR1 64/4885CNR2 24/4885
US-20040235855-A1 Phospholipase C inhibitors for use in treating inflammatory disorders PLA2G4C, PLA2G4B, PLA2G5 KMT2A 4455/4885CNR1 141/4885CNR2 105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.