SCHEMBL6687345

SCHEMBL6687345

COc1cccc(C(=O)NCCC(C(=O)NCCC2CNc3ccc(F)cc32)C2CCCCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.45
DRD4 P21917 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CTSL P07711 8/20 0.41
CTSK P43235 3/20 0.41
HDAC8 Q9BY41 1/20 0.40
CCR3 P51677 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690325 0.95 CTSS (0.46) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6689425 0.94 HDAC8 (0.42) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6687213 0.90 RAB9A (0.41) CTSSNPC1RAB9ASMN1; SMN2CTSL
SCHEMBL6690013 0.87 CCR3 (0.40) CTSSCTSLCTSKHDAC8CCR3
SCHEMBL6690556 0.87 CTSS (0.43) CTSSNPC1RAB9ASMN1; SMN2CTSL
SCHEMBL6693415 0.86 MEN1 (0.41) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6691059 0.86 ALDH1A1 (0.41) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6698515 0.84 DRD4 (0.39) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6693429 0.84 DRD4 (0.39) CTSSDRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6691040 0.83 CTSS (0.44) CTSSDRD4CTSLCTSKHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed