SCHEMBL6690556

SCHEMBL6690556

COc1cccc(C(=O)NCCC(C(=O)NCCC2CNc3c(F)cccc32)C2CCCCC2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.43
CTSL P07711 5/20 0.41
CTSK P43235 2/20 0.41
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
RAB9A P51151 4/20 0.39
NPC1 O15118 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
GAA P10253 2/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6691059 0.92 ALDH1A1 (0.41) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6690325 0.88 CTSS (0.46) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6687345 0.87 CTSS (0.45) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6689425 0.87 HDAC8 (0.42) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6687213 0.83 RAB9A (0.41) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6693415 0.82 MEN1 (0.41) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6690013 0.81 CCR3 (0.40) CTSSCTSLCTSKALDH1A1MEN1
SCHEMBL6690007 0.74 CTSS (0.65) CTSSCTSLCTSK
SCHEMBL6691086 0.72 CTSS (0.59) CTSSCTSLCTSK
SCHEMBL6691040 0.72 CTSS (0.44) CTSSCTSLCTSKALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed