SCHEMBL6689425

SCHEMBL6689425

COc1cccc(C(=O)NCCC(C(=O)NCCC2CNc3ccc(OC)cc32)C2CCCCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.42
CTSL P07711 3/20 0.42
CTSS P25774 3/20 0.42
CTSK P43235 1/20 0.42
ALDH1A1 P00352 4/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 2/20 0.42
MAPT P10636 1/20 0.42
NQO2 P16083 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
DRD4 P21917 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687345 0.94 CTSS (0.45) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6690013 0.93 CCR3 (0.40) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6687213 0.93 RAB9A (0.41) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6690325 0.90 CTSS (0.46) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6693415 0.88 MEN1 (0.41) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6691059 0.88 ALDH1A1 (0.41) CTSLCTSSCTSKALDH1A1MEN1
SCHEMBL6690556 0.87 CTSS (0.43) CTSLCTSSCTSKALDH1A1MEN1
SCHEMBL6698515 0.78 DRD4 (0.39) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6693429 0.78 DRD4 (0.39) HDAC8CTSLCTSSCTSKALDH1A1
SCHEMBL6690876 0.77 DRD4 (0.38) HDAC8CTSLCTSSCTSKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed