SCHEMBL6687902

SCHEMBL6687902

[CH]1C=CC(N2CCC(N3CCCCC3)CC2)=CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 13/20 0.47
L3MBTL1 Q9Y468 12/20 0.47
MBTD1 Q05BQ5 7/20 0.44
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
TP53BP1 Q12888 3/20 0.36
L3MBTL4 Q8NA19 2/20 0.36
HRH3 Q9Y5N1 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2479690 0.85 HRH3 (0.34) L3MBTL3L3MBTL1MBTD1HRH3
SCHEMBL2480855 0.85 HRH3 (0.34) L3MBTL3L3MBTL1HRH3
SCHEMBL695794 0.82 ALDH1A1 (0.31)
SCHEMBL1900342 0.82 ALDH1A1 (0.31)
SCHEMBL188370 0.77
SCHEMBL1681276 0.76 TSHR (0.37) L3MBTL1HRH3
SCHEMBL18403928 0.70 L3MBTL3 (0.46) L3MBTL3L3MBTL1MBTD1CYP2D6CYP2C19
SCHEMBL187983 0.68 ADRB1 (0.36)
SCHEMBL2480196 0.68 FAAH (0.32) L3MBTL3L3MBTL1
SCHEMBL2483385 0.68 CASP1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004083173-A2 KETOPIPERAZINE DERIVATIVES AS BRADYKININ ANTAGONISTS MERCK & CO., INC. (US) 2004-09-30 WO disclosed