SCHEMBL6688055

SCHEMBL6688055

CC(C)(C)OC(=O)Nc1ccc(/C=C/C2CC(=O)N2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
PSMB8 P28062 1/20 0.38
NPC1 O15118 1/20 0.38
F13A1 P00488 1/20 0.38
TGM2 P21980 1/20 0.38
TGM1 P22735 1/20 0.38
CYP17A1 P05093 2/20 0.37
PRKDC P78527 1/20 0.37
DRD2 P14416 1/20 0.36
LIPE Q05469 1/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6688061 1.00 HDAC1 (0.40) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6685062 0.87 HDAC3 (0.44) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6685056 0.87 HDAC3 (0.44) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6685069 0.87 HDAC3 (0.44) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6690143 0.84 GPR119 (0.41) HDAC1PTPN1NPC1
SCHEMBL6690141 0.84 GPR119 (0.41) HDAC1PTPN1NPC1
SCHEMBL6687262 0.82 ALDH1A1 (0.43) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6687260 0.82 ALDH1A1 (0.43) HDAC1HDAC3HDAC2HDAC8HDAC6
SCHEMBL6687420 0.80 LMNA (0.47) PTPN1
SCHEMBL6687419 0.80 LMNA (0.47) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004089362-A1 2-CYANOPYRROLES AND THEIR ANALOGUES AS DDP-IV INHIBITORS NOVO NORDISK A/S (DK) 2004-10-21 WO disclosed