Heteronium

Heteronium

SCHEMBL668862

C[N+]1(C)CCC(OC(=O)C(O)(c2ccccc2)c2cccs2)C1.[Br-]

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Heteronium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM3 known ✓ P20309 17/20 0.66
CHRM2 known ✓ P08172 15/20 0.66
CHRM1 known ✓ P11229 8/20 0.59
CHRM4 known ✓ P08173 1/20 0.59
CHRM5 known ✓ P08912 1/20 0.59
SLC22A1 O15245 1/20 0.66
KCNH2 Q12809 2/20 0.64
LMNA P02545 1/20 0.64
CYP2D6 P10635 1/20 0.64
CYP2C19 P33261 1/20 0.64
SLC6A4 P31645 1/20 0.64
HRH1 P35367 1/20 0.59
HTR2B P41595 1/20 0.59
RAB9A P51151 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Heteronium SCHEMBL249397 0.99 CHRM3 (0.65) CHRM3CHRM2SLC22A1KCNH2LMNA
Benzopyrronium SCHEMBL916243 0.87 CHRM3 (0.85) CHRM3CHRM2SLC22A1KCNH2LMNA
Benzopyrronium SCHEMBL2111041 0.86 CHRM3 (0.85) CHRM3CHRM2SLC22A1KCNH2LMNA
Parapenzolate SCHEMBL636125 0.81 CHRM3 (0.74) CHRM3CHRM2SLC22A1KCNH2LMNA
Bromide SCHEMBL11483400 0.81 CHRM3 (0.50) CHRM3CHRM2SLC22A1KCNH2LMNA
Bromide SCHEMBL131394 0.80 CHRM3 (0.69) CHRM3CHRM2SLC22A1KCNH2CHRM1
Bromide SCHEMBL130614 0.80 CHRM3 (0.69) CHRM3CHRM2SLC22A1KCNH2CHRM1
Mepenzolate SCHEMBL15575981 0.80 CHRM3 (1.00) CHRM3CHRM2SLC22A1KCNH2LMNA
Mepenzolate SCHEMBL99030 0.80 CHRM3 (1.00) CHRM3CHRM2SLC22A1KCNH2LMNA
Mepenzolate SCHEMBL147471 0.80 CHRM3 (1.00) CHRM3CHRM2SLC22A1KCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 328 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140171645-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE HOVIONE INTER LTD. (CH) 2014-06-19 US claimed
EP-2691367-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE Hovione Inter Ltd. (CH) 2014-02-05 EP claimed
CN-103502211-A Electrophilic alkylating reagents, preparation and use thereof HOVIONE FARMACIENCIA S A 2014-01-08 CN claimed
WO-2012131286-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE HOVIONE INTER. LTD (CH) 2012-10-04 WO claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5008111-A Pretreating skin with anticholinergic quaternary ammonium salt to suppress perspiration SCHERING CORPORATION (US) 1991-04-16 US claimed
US-4824676-A ANTICHOLINERGIC AGENT TO SUPPRESS PERSPIRATION SCHERING CORPORATION (US) 1989-04-25 US claimed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
WO-1997040034-A1 SOLID PHASE AND COMBINATORIAL SYNTHESIS OF SUBSTITUTED THIOPHENES AND OF ARRAYS OF SUBSTITUTED THIOPHENES NOVO NORDISK A/S (DK) 1997-10-30 WO disclosed
US-5656286-A BLEND OF TWO POLYMERS; PRESSURE SENSITIVE ADHESIVE NOVEN PHARMACEUTICALS, INC. (US) 1997-08-12 US disclosed
WO-1996040084-A1 COMPOSITIONS AND METHODS FOR USE OF PRESSURE SENSITIVE ADHESIVE TRANSDERMAL DEVICES CONTAINING A BIOADHESIVE HUMECTANT NOVEN PHARMACEUTICALS, INC. (US) 1996-12-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES SORD, SLC6A13, CACNA1A CHRM3 560/4885CHRM2 158/4885CHRM1 312/4885
US-20140171645-A1 ELECTROPHILIC ALKYLATING REAGENTS, THEIR PREPARATION AND USE MGMT, MCL1, TOP2B CHRM3 3125/4885CHRM2 2607/4885CHRM1 3157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.