SCHEMBL6688950

SCHEMBL6688950

CCNC(=NC(=O)OC(C)(C)C)Nc1cccc(CN(C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.42
AOC3 Q16853 5/20 0.39
RIPK1 Q13546 3/20 0.38
HTR2C P28335 1/20 0.37
SLC6A4 P31645 1/20 0.37
MCHR1 Q99705 1/20 0.36
BACE1 P56817 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678217 0.91 KDM1A (0.40) AOC3RIPK1SMN1; SMN2MEN1NPC1
SCHEMBL6685806 0.88 ACHE (0.43) BACE1SMN1; SMN2MEN1KMT2A
SCHEMBL6681938 0.82 HTT (0.39) MCHR1SMN1; SMN2MEN1GAAMAPT
SCHEMBL6674967 0.80 GRM2 (0.38) GLSAOC3BACE1SMN1; SMN2MEN1
SCHEMBL7247906 0.80 LMNA (0.34) GLSRIPK1HTR2CSLC6A4MCHR1
SCHEMBL6679118 0.79 SENP1 (0.49) SMN1; SMN2MAPTRAB9A
SCHEMBL6685809 0.78 KMT2A (0.41) SMN1; SMN2MEN1NPC1MAPTRAB9A
SCHEMBL6682104 0.78 HDAC3 (0.35) GLSBACE1MEN1RAB9AKMT2A
SCHEMBL7238099 0.77 GLS (0.46) GLSAOC3HTR2CSLC6A4BACE1
SCHEMBL6679942 0.77 MCHR1 (0.32) MCHR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed