SCHEMBL6689803

SCHEMBL6689803

COc1cccc(C(=O)NCCC(C)(C)CC(=O)N(CCC2CNc3ccc(F)cc32)COCc2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.39
DRD4 P21917 3/20 0.37
MAPT P10636 1/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CCR3 P51677 1/20 0.36
ACHE P22303 1/20 0.35
CTSD P07339 1/20 0.35
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689978 0.86 SIGMAR1 (0.33) SIGMAR1RAB9ACTSLCTSS
SCHEMBL6689430 0.82 CTSS (0.37) SIGMAR1DRD4MAPTNPC1RAB9A
SCHEMBL6693989 0.81 CTSS (0.41) NPC1RAB9AMEN1KMT2ACTSL
SCHEMBL6688100 0.81 CTSS (0.41) SIGMAR1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL6688064 0.73 CTSS (0.42) SIGMAR1DRD4NPC1RAB9ASMN1; SMN2
SCHEMBL6693429 0.68 DRD4 (0.39) DRD4MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL6690876 0.67 DRD4 (0.38) SIGMAR1DRD4MAPTNPC1RAB9A
SCHEMBL8286606 0.66 IDO1 (0.53) MAPTSMN1; SMN2MEN1KMT2ACTSL
SCHEMBL6690013 0.65 CCR3 (0.40) SIGMAR1MEN1KMT2ACTSLCTSS
SCHEMBL6698515 0.65 DRD4 (0.39) DRD4MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed