SCHEMBL6689430

SCHEMBL6689430

COc1cccc(C(=O)NC[C@H](C(=O)N(CCC2CNc3ccc(F)cc32)COCc2ccccc2)c2ccc(F)cc2)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.37
CTSL P07711 2/20 0.37
SIGMAR1 Q99720 1/20 0.36
DRD4 P21917 1/20 0.36
MAPT P10636 2/20 0.36
CTSK P43235 1/20 0.36
TP53 P04637 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
GPR139 Q6DWJ6 2/20 0.34
OPRM1 P35372 1/20 0.34
CCR3 P51677 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693989 0.89 CTSS (0.41) CTSSCTSLCTSKNPC1RAB9A
SCHEMBL6688100 0.88 CTSS (0.41) CTSSCTSLSIGMAR1CTSKNPC1
SCHEMBL6689803 0.82 SIGMAR1 (0.39) CTSSCTSLSIGMAR1DRD4MAPT
SCHEMBL6688064 0.73 CTSS (0.42) CTSSCTSLSIGMAR1DRD4CTSK
SCHEMBL6689978 0.69 SIGMAR1 (0.33) CTSSCTSLSIGMAR1RAB9A
SCHEMBL6693429 0.68 DRD4 (0.39) CTSSCTSLDRD4MAPTCTSK
SCHEMBL6690876 0.68 DRD4 (0.38) CTSSCTSLSIGMAR1DRD4MAPT
SCHEMBL6687345 0.67 CTSS (0.45) CTSSCTSLDRD4CTSKNPC1
SCHEMBL4799699 0.67 CTSS (0.55) CTSSCTSLCTSK
SCHEMBL6698515 0.66 DRD4 (0.39) CTSSCTSLDRD4MAPTCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed