SCHEMBL6690522

SCHEMBL6690522

CCOc1ccc(NC(=N)N[N+](=O)[O-])cc1CNC(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
PTPN1 P18031 6/20 0.36
RORC P51449 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTPN2 P17706 4/20 0.35
PTPN11 Q06124 2/20 0.35
PTPN6 P29350 2/20 0.35
PTPRF P10586 1/20 0.35
POLB P06746 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
PRMT1 Q99873 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NAMPT P43490 1/20 0.34
NPBWR1 P48145 1/20 0.34
MCHR1 Q99705 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
KCNB1 Q14721 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246439 0.90 ALDH1A1 (0.43) ALDH1A1PTPN11POLBMEN1KMT2A
SCHEMBL6681426 0.88 CYP2C9 (0.42) ALDH1A1TDP1POLBMEN1KMT2A
SCHEMBL6690531 0.82 ALDH1A1 (0.39) ALDH1A1PTPN1RORCTDP1PTPN2
SCHEMBL6676307 0.80 NAMPT (0.52) TDP1PTPN11MAPTPRMT1GAA
SCHEMBL6678283 0.80 TDP1 (0.42) ALDH1A1RORCTDP1POLBMEN1
SCHEMBL6677097 0.79 ALDH1A1 (0.46) ALDH1A1PTPN1RORCTDP1PTPN2
Hydrochloric Acid SCHEMBL6680091 0.79 TDP1 (0.41) ALDH1A1RORCTDP1POLBMEN1
SCHEMBL6676086 0.79 NPBWR1 (0.54) ALDH1A1POLBMEN1KMT2AMAPT
SCHEMBL6679736 0.79 GLS (0.46) MEN1KMT2AMAPTNAMPT
SCHEMBL6674829 0.76 PTPN1 (0.38) ALDH1A1PTPN1RORCTDP1PTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed