SCHEMBL6691067

SCHEMBL6691067

COc1c(C)cc(NCCN(C(N)=O)C(=O)[CH]CC2CCCCC2)cc1C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CNR1 P21554 3/20 0.35
CNR2 P34972 3/20 0.35
KMT2A Q03164 3/20 0.34
METAP2 P50579 3/20 0.33
MEN1 O00255 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
EPHX2 P34913 1/20 0.32
PARP15 Q460N3 1/20 0.31
PARP10 Q53GL7 1/20 0.31
CTSL P07711 3/20 0.31
CTSS P25774 3/20 0.31
CTSK P43235 2/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5409955 0.83 EPHX2 (0.47) ALDH1A1EPHX2CTSLCTSSCTSK
SCHEMBL6693494 0.83 SLC6A9 (0.37) PARP10RAB9A
SCHEMBL5404160 0.82 EPHX2 (0.46) ALDH1A1EPHX2CTSLCTSSCTSK
SCHEMBL6685923 0.78 RAB9A (0.38) CTSLCTSSCTSKRAB9A
SCHEMBL6693491 0.77 NPC1 (0.42) ALDH1A1TDP1KMT2AMEN1EPHX2
SCHEMBL6688679 0.77 NPC1 (0.39) ALDH1A1TDP1KMT2AMEN1EPHX2
SCHEMBL6688042 0.76 HTR7 (0.39) ALDH1A1TDP1KMT2AMEN1PARP15
SCHEMBL6693564 0.76 CDK1 (0.37) PARP15PARP10CTSS
SCHEMBL6690542 0.76 RORC (0.41) ALDH1A1KMT2AMEN1NPSR1
SCHEMBL6685681 0.76 EPHX2 (0.48) ALDH1A1CNR2KMT2AMETAP2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed