SCHEMBL6694701

SCHEMBL6694701

CC(=O)N1CCC(C(CC2NC(=O)NC2=O)NC(=O)c2ccc(COc3cccc4ncccc34)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.39
IDO1 P14902 3/20 0.38
CYP3A4 P08684 2/20 0.38
GCK P35557 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CASP1 P29466 1/20 0.35
CASP3 P42574 1/20 0.35
CASP7 P55210 1/20 0.35
CASP8 Q14790 1/20 0.35
HTR1A P08908 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050275 0.87 CHRM2 (0.40) CHRM2IDO1CYP3A4GCKSMN1; SMN2
SCHEMBL6692739 0.84 MEN1 (0.40) IDO1SMN1; SMN2ALDH1A1MAPTHDAC6
SCHEMBL6694703 0.83 P2RX7 (0.37) CHRM2GCKSMN1; SMN2HTR1AALDH1A1
SCHEMBL6694698 0.79 SMN1; SMN2 (0.36) CHRM2GCKSMN1; SMN2HTR1AALDH1A1
SCHEMBL6700685 0.78 MEN1 (0.41) MAPTKDM4E
SCHEMBL4050732 0.75 RAB9A (0.38) CASP1CASP3CASP7CASP8ALDH1A1
SCHEMBL6677177 0.71 MMP12 (0.59)
SCHEMBL4048796 0.71 MEN1 (0.41) SMN1; SMN2ALDH1A1MAPTHDAC6KDM4E
SCHEMBL6692741 0.67 HDAC6 (0.40) SMN1; SMN2ALDH1A1MAPTHDAC6KDM4E
SCHEMBL8739476 0.67 EZH2 (0.63) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397137-A4 HYDANTION DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES BRISTOL MYERS SQUIBB CO (US) 2004-10-13 EP disclosed
EP-1397137-A1 HYDANTION DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2004-03-17 EP disclosed
WO-2002096426-A1 HYDANTION DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-12-05 WO disclosed