Bromide

Bromide

SCHEMBL6697756

Br.Clc1cccc[n+]1Cc1ccccc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 3/20 0.38
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
KDM4E B2RXH2 3/20 0.42
HTT P42858 3/20 0.42
HPGD P15428 2/20 0.42
NPC1 O15118 1/20 0.42
MITF O75030 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
BCHE P06276 1/20 0.38
LMNA P02545 4/20 0.36
CHKA P35790 3/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31130749 0.98 CYP2D6 (0.47) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
SCHEMBL6162141 0.98 CYP2D6 (0.47) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
Bromide SCHEMBL571679 0.96 CYP2D6 (0.46) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
SCHEMBL10333361 0.84 CYP2D6 (0.39) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
SCHEMBL25262661 0.82 KDM4E (0.42) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
SCHEMBL25282130 0.78 ACHE (0.49) ALDH1A1SMN1; SMN2KDM4EHTTNPC1
Bromide SCHEMBL11799324 0.76 ALDH1A1 (0.37) CYP2D6CYP2C19ALDH1A1SMN1; SMN2HPGD
Benzene SCHEMBL9542509 0.74 KDM4E (0.42) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E
SCHEMBL19504336 0.73 MAOA (0.40) KDM4ELMNACHKACHKB
Hydrochloric Acid SCHEMBL11363136 0.72 KDM4E (0.47) CYP2D6CYP2C19ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040138284-A1 Indol-3-yl derivatives WIESNER MATTHIAS 2004-07-15 US disclosed
US-6743810-B2 INTEGRIN INHIBITORS; TUMORS, OSTEOPOROSIS, OSTEOLYTIC DISEASES, SUPPRESSING ANGIOGENESIS, ANTITHROMBOTIC MERCK PATENT GMBH (DE) 2004-06-01 US disclosed
US-20030045728-A1 Liberating 3-substituted indole compound from one of its functional derivatives by treatment with a solvolyzing or hydrogenating agent, amidation, saponification, alkylation or acylation, or salt formation MERCK PATENT GMBH (DE) 2003-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030045728-A1 Liberating 3-substituted indole compound from one of its functional derivatives by treatment with a solvolyzing or hydrogenating agent, amidation, saponification, alkylation or acylation, or salt formation IGF1R, IDO1, ITGB3 ACHE 1246/4885CYP2D6 3223/4885CYP2C19 3396/4885
US-20040138284-A1 Indol-3-yl derivatives ITGB3, ITGB1, IGF1R ACHE 1596/4885CYP2D6 3475/4885CYP2C19 3546/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.