SCHEMBL6698

SCHEMBL6698

COc1cccc(SC(CO)c2c(C)noc2-c2ccc(Br)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MTNR1A P48039 9/20 0.36
MTNR1B P49286 9/20 0.36
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAOB P27338 1/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
BRD4 O60885 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387 0.85 NR1I2 (0.35) RAB9ATDP1L3MBTL1BRD4SMN1; SMN2
SCHEMBL6652 0.83 MEN1 (0.38) MEN1KMT2AMTNR1AMTNR1BHPGD
SCHEMBL6697 0.82 MTNR1A (0.40) MEN1KMT2AMTNR1AMTNR1BHPGD
SCHEMBL6651 0.74 MAPT (0.41) MEN1KMT2AMTNR1AMTNR1BHPGD
SCHEMBL11802 0.74 CYP1A2 (0.33) RAB9AHTTTDP1SMN1; SMN2MAPT
SCHEMBL6943 0.72 EPHX1 (0.35) RAB9AL3MBTL1SMN1; SMN2MAPTALDH1A1
SCHEMBL2087 0.72 EPHX1 (0.35) RAB9AL3MBTL1SMN1; SMN2MAPTALDH1A1
SCHEMBL2762295 0.72 FPR2 (0.40) MEN1KMT2AHPGDRAB9AHTT
SCHEMBL6814 0.71 CYP1A2 (0.31) TDP1
SCHEMBL1627 0.70 EPHX1 (0.41) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed