SCHEMBL6703290

SCHEMBL6703290

CN1C(=O)N(Cc2ccc(C(=O)O)cc2)Cc2nc(C#CCc3ccccc3)oc21

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 5/20 0.43
SLC22A8 Q8TCC7 1/20 0.43
HDAC6 Q9UBN7 5/20 0.37
AGTR1 P30556 3/20 0.35
AGTR2 P50052 3/20 0.35
XIAP P98170 1/20 0.34
BIRC2 Q13490 1/20 0.34
PTGER4 P35408 1/20 0.34
PPARG P37231 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
HDAC1 Q13547 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6699862 0.93 MMP13 (0.36) MMP13SLC22A8AGTR1AGTR2PTGER4
SCHEMBL6920079 0.89 MMP13 (0.38) MMP13SLC22A8HDAC6AGTR1AGTR2
SCHEMBL6289326 0.85 MMP13 (0.43) MMP13SLC22A8HDAC6AGTR1AGTR2
SCHEMBL6694967 0.81 MMP13 (0.46) MMP13SLC22A8HDAC6SLC6A3
SCHEMBL6696978 0.79 PTGER4 (0.46) MMP13HDAC6PTGER4
SCHEMBL6701922 0.78 SCD (0.36) MMP13SLC22A8AGTR1AGTR2PTGER4
SCHEMBL6289360 0.76 MMP13 (0.46) MMP13SLC22A8HDAC6HDAC1HDAC8
SCHEMBL6706890 0.73 MMP13 (0.55) MMP13SLC22A8HDAC6HDAC1HDAC8
SCHEMBL6292726 0.72 MMP13 (0.46) MMP13SLC22A8HDAC6HDAC1HDAC8
SCHEMBL5189013 0.69 HDAC6 (0.50) HDAC6HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040038994-A1 Pyrimidine fused bicyclic metalloproteinase inhibitors WILSON MICHAEL WILLIAM (US) 2004-02-26 US disclosed
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038994-A1 Pyrimidine fused bicyclic metalloproteinase inhibitors MMP9, MMP1, MMP2 MMP13 13/4885SLC22A8 2959/4885HDAC6 493/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.