SCHEMBL6706934

SCHEMBL6706934

CC(O)C(C)(NCc1ccc(OCc2ccc(SC(F)(F)F)cc2)c([N+](=O)[O-])c1)C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 9/20 0.41
CD274 Q9NZQ7 9/20 0.41
CTSV O60911 2/20 0.38
CTSL P07711 2/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 4/20 0.37
ALDH1A1 P00352 1/20 0.36
ALPG P10696 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
PTPRZ1 P23471 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6688691 0.84 PDCD1 (0.44) PDCD1CD274CTSVCTSLLMNA
SCHEMBL6694008 0.82 PDCD1 (0.44) PDCD1CD274CTSVCTSLLMNA
SCHEMBL6706928 0.79 PDCD1 (0.51) PDCD1CD274CTSVCTSLMAPT
SCHEMBL6235743 0.73 PDCD1 (0.39) PDCD1CD274CTSVCTSLLMNA
SCHEMBL13959005 0.72 PDCD1 (0.50) PDCD1CD274CTSVCTSLLMNA
SCHEMBL6234734 0.71 ALDH1A1 (0.48) PDCD1CD274CTSVCTSLLMNA
SCHEMBL6232647 0.69 PDCD1 (0.41) PDCD1CD274CTSVCTSLLMNA
SCHEMBL6685864 0.69 MAOB (0.46) CD274PTPRZ1
SCHEMBL6685862 0.69 MAOB (0.46) CD274PTPRZ1
SCHEMBL6693067 0.69 MAOB (0.45) PDCD1CD274ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed