SCHEMBL6709937

SCHEMBL6709937

COC[C@@H]1C2CN(c3ccc(F)cc3NC(=O)OCc3ccccc3)C[C@@H]21

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 10/20 0.46
MGAT2 Q10469 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KDM1A O60341 5/20 0.43
MAOA P21397 5/20 0.43
KDM1B Q8NB78 5/20 0.43
RCOR1 Q9UKL0 5/20 0.43
MAOB P27338 3/20 0.42
MGLL Q99685 1/20 0.42
CASP3 P42574 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6338415 0.85 MAPT (0.45) NPC1RAB9AKDM1AMAOARCOR1
SCHEMBL6712840 0.83 MGAT2 (0.42) CHRM3MGAT2KDM1AMAOAKDM1B
SCHEMBL6709795 0.81 MGAT2 (0.41) CHRM3MGAT2NPC1RAB9AKDM1A
SCHEMBL5746506 0.78 RORC (0.42) CHRM3MGAT2NPC1RAB9AKDM1A
SCHEMBL285633 0.73 RAB9A (0.60) MGAT2NPC1RAB9AMAOBMGLL
SCHEMBL524207 0.71 SMN1; SMN2 (0.52) NPC1RAB9A
SCHEMBL524206 0.71 SMN1; SMN2 (0.52) NPC1RAB9A
SCHEMBL28355514 0.71 MGLL (0.55) MGAT2NPC1RAB9AMAOBMGLL
SCHEMBL30207791 0.71 MGLL (0.55) NPC1RAB9AMAOBMGLLCASP3
SCHEMBL6711214 0.70 MGAT2 (0.37) CHRM3MGAT2NPC1RAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385834-A1 BICYCLO[3,1,0]HEXANE CONTAINING OXAZOLIDINONE ANTIBIOTIC AND DERIVATIVES THEREOF Merck & Co., Inc. (US) 2004-02-04 EP disclosed
WO-2003027083-A1 BICYCLO[3,1,0]HEXANE CONTAINING OXAZOLIDINONE ANTIBIOTIC AND DERIVATIVES THEREOF MERCK & CO., INC. (US) 2003-04-03 WO disclosed