SCHEMBL6714654

SCHEMBL6714654

CCc1[nH]c2cc(Cl)c(F)cc2c(=O)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.39
TDO2 P48775 3/20 0.39
GPR84 Q9NQS5 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
MAP2 P11137 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5716984 0.82 ALOX5 (0.41) PTGS1PTGS2MAP2PIM1PIM2
SCHEMBL11204197 0.79 IDO1 (0.38) IDO1TDO2GPR84PTGS1PTGS2
SCHEMBL11203471 0.79 GPR84 (0.38) IDO1TDO2GPR84PTGS1PTGS2
SCHEMBL3474228 0.77 ALDH1A1 (0.53) KDM4EALDH1A1
SCHEMBL9877122 0.76 KCNH2 (0.36) IDO1TDO2KDM4EALDH1A1
SCHEMBL6904417 0.75 IDO1 (0.38) IDO1TDO2GPR84PTGS1PTGS2
SCHEMBL8959621 0.74 PRNP (0.55) PTGS1PTGS2MAP2
SCHEMBL10974102 0.73 NPC1 (0.43) KDM4EALDH1A1
SCHEMBL5716973 0.73 ALOX5 (0.58)
SCHEMBL7008377 0.72 PRKAB2 (0.42) PTGS1PTGS2PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401829-A4 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX INC (US) 2004-10-27 EP disclosed
EP-1453846-A1 MACROLIDES GLAXO GROUP LIMITED (GB) 2004-09-08 EP disclosed
EP-1401829-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS Microbiotix, Inc. (US) 2004-03-31 EP disclosed
WO-2003042228-A1 MACROLIDES GLAXO GROUP LIMITED (GB) 2003-05-22 WO disclosed
WO-2002102792-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX, INC. (US) 2002-12-27 WO disclosed