SCHEMBL6748926

SCHEMBL6748926

COc1ccc(-c2oc3cc(OC)ccc3c2-c2cc(OCCN(C)C)ccc2C=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.49
BCHE P06276 3/20 0.46
ACHE P22303 3/20 0.46
SIGMAR1 Q99720 2/20 0.45
HRH3 Q9Y5N1 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALK Q9UM73 2/20 0.42
RAB9A P51151 1/20 0.41
KDR P35968 1/20 0.40
TOP1 P11387 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6748797 0.91 BCHE (0.58) BCHEACHEHRH3MAPTKMT2A
SCHEMBL6747002 0.90 BCHE (0.43) ESR1BCHEACHEHRH3KDM4E
SCHEMBL7117346 0.88 ALDH1A1 (0.53) BCHEACHEKDM4EMEN1ALDH1A1
SCHEMBL8589084 0.86 ESR1 (0.50) ESR1BCHEACHESIGMAR1HRH3
SCHEMBL6749914 0.83 BCHE (0.58) ESR1BCHEACHEHRH3KDM4E
SCHEMBL5924015 0.80 MAPT (0.56) BCHEACHEKDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL6746980 0.77 ESR1 (0.51) ESR1BCHEACHEHRH3ALK
SCHEMBL6744872 0.76 ESR1 (0.52) ESR1BCHEACHESIGMAR1HRH3
Hydrochloric Acid SCHEMBL8589257 0.75 BCHE (0.43) ESR1BCHEACHEHRH3KDM4E
Hydrochloric Acid SCHEMBL6744836 0.75 ESR1 (0.51) ESR1BCHEACHESIGMAR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6703407-B1 TREATMENT OF MENOPAUSAL SYNDROME, UTERINE FIBROID DISEASE, ENDOMETRIOSIS, AND AORTAL SMOOTH MUSCLE CELL PROLIFERATION ELI LILLY AND COMPANY 2004-03-09 US disclosed
EP-0774966-B1 BENZOFURAN COMPOUNDS, COMPOSITIONS, AND METHODS LILLY CO ELI (US) 2003-11-05 EP disclosed
EP-0774966-A4 BENZOFURAN COMPOUNDS, COMPOSITIONS, AND METHODS LILLY CO ELI (US) 1998-01-07 EP disclosed
EP-0774966-A1 BENZOFURAN COMPOUNDS, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1997-05-28 EP disclosed
WO-1996009040-A1 BENZOFURAN COMPOUNDS, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1996-03-28 WO disclosed